Patent · US Expired

Chemical compounds

US5714148A · kind A · utility

4Cited by
1References
21Claims
0Family size

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Inventors

Key dates

Filing dateSep 30, 1996
Grant dateFeb 3, 1998
Priority date
Expiry dateSep 30, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C311/51
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Prodrugs, of generic formula I, are disclosed for use in antibody directed enzyme prodrug therapy (ADEPT). The prodrugs are substrates for carboxypeptidase G2 (CPG2) and yield more active cytotoxic drugs than known products of CPG2 catalysed reactions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.