Patent · US Expired

Isoxazoline compounds as antiinflammatory agents

US5716967A · kind A · utility

40Cited by
5References
16Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 15, 1996
Grant dateFeb 10, 1998
Priority date
Expiry dateMay 15, 2016

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

This invention relates to isoxazoline compounds which are selective inhibitors of phosphodiesterase type IV (PDE.sub.IV). The isoxazoline compounds are useful in inhibiting PDE.sub.IV and in the treatment of AIDS, asthma, arthritis, bronchitis, chronic obstructive pulmonary disease, psoriasis, allergic rhinitis, dermatitis, shock, atopic dermatitis, rheumatoid arthritis and osteoarthritis. This invention also relates to pharmaceutical compositions useful therefor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.