Patent · US Expired

6-membered ring fused imidazoles as muscarinic agents

US5723468A · kind A · utility

0Cited by
2References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 1, 1996
Grant dateMar 3, 1998
Priority date
Expiry dateOct 1, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D453/02
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The compound of the formula: ##STR1## where R.sub.1 is H, alkyl, perhaloalkyl, arylalkyl, alkenyl or alkynyl; R.sub.2 is H when R.sub.4 is other than H, and, when R.sub.4 is H, R.sub.2 is ##STR2## in which R.sub.5 is hydrogen or alkyl; R.sub.3 is hydrogen or halogen; R.sub.4 is H or ##STR3## X and Y are nitrogen and Z is carbon; n is 1 or 2; n.sub.1 is 0, 1, 2, 3, 4, or 5; or a pharmaceutically acceptable salt thereof are centrally active muscarinic agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.