Patent · US Expired

Methods for preparing antiproliferative 5-substituted pyrimidone compounds

US5726312A · kind A · utility

3Cited by
8References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 24, 1995
Grant dateMar 10, 1998
Priority date
Expiry dateMay 24, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Intermediates for preparing derivatives of 5-thia- and 5-selenopyrimidinone, ##STR1## which are useful as inhibitors of the enzymes glycinamide ribonucleotide formyl transferase (GARFT) and amino imidazole carboxamide ribonucleotide formyl transferase (AICARFT). The present invention is also directed to methods of preparing these intermediates.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.