Patent · US Expired

Hypoxanthine and guanine compounds

US5736549A · kind A · utility

25Cited by
2References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 5, 1995
Grant dateApr 7, 1998
Priority date
Expiry dateOct 5, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D473/18
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of formula I ##STR1## where n=0-2; PA1 R.sup.1 is H, NH.sub.2 or a halogen; PA1 R.sup.2 is H or NH.sub.2 ; PA1 R.sup.3 is any of the four groups ##STR2## where m=0 or 1; and PA1 X is O, NR.sup.5, or S(O).sub.0-2 and, in group (b), the X's may be the same or different. Compounds of the invention have utility as inhibitors of purine nucleoside phosphyorylase (PNP).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.