Patent · US Expired

Cannabinoid receptor antagonists

US5747524A · kind A · utility

50Cited by
11References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 30, 1996
Grant dateMay 5, 1998
Priority date
Expiry dateSep 30, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D307/88
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

This invention discloses methods of using certain aryl-benzob!thiophene and benzob!furan compounds to block or inhibit cannabinoid receptors in mammals. It also discloses novel compounds which are antagonists of the cannabinoid receptors and also discloses pharmaceutical formulations which contain the compounds as an active ingredient.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.