Patent · US Expired

Bicyclopolyazamacrocyclophosphonic acid half esters

US5750660A · kind A · utility

19Cited by
27References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 15, 1996
Grant dateMay 12, 1998
Priority date
Expiry dateJul 15, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/6561
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Bicyclopolyazamacrocyclophosphonic acid compounds are disclosed which may form inert complexes with Gd, Mn or Fe ions. The overall charge of the complex can be varied to alter the in vivo biolocalization. Such complexes can be covalently attached to an antibody, antibody fragment or other biologically active molecule to form conjugates. The complexes and conjugates are useful as contrast agents for diagnostic purposes.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.