Patent · US Expired

Method of preparing certain 3-halo-imidazopyridines

US5750699A · kind A · utility

24Cited by
0References
1Claims
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Assignee

Inventors

Key dates

Filing dateJun 12, 1996
Grant dateMay 12, 1998
Priority date
Expiry dateJun 12, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to bradykinin antagonists of the formula: ##STR1## wherein R.sup.1 is halogen, PA1 R.sup.2 and R.sup.3 are each hydrogen, lower alkyl, halo(lower)alkyl or acyl, PA1 R.sup.4 is aryl having suitable substituent(s), or a heterocyclic group optionally having suitable substituent(s), PA1 Q is O or N--R.sup.11, in which R.sup.11 is hydrogen or acyl, and PA1 A is lower alkylene, and pharmaceutically acceptable salts thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.