Patent · US Expired

Biphenysulfonamide matrix metal alloproteinase inhibitors

US5756545A · kind A · utility

19Cited by
7References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 21, 1997
Grant dateMay 26, 1998
Priority date
Expiry dateApr 21, 2017

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/195
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## wherein R.sup.1 includes alkyl, halo, nitro, amino, cyano, alkoxy, and alkoxycarbonyl; R.sup.2 is alkyl and substituted alkyl; and R.sup.3 is OH or NHOH are useful for inhibiting matrix metalloproteinase enzymes in animals, and as such, prevent and treat diseases resulting from the breakdown of connective tissues.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.