Patent · US Expired

Combinatorial process for synthesizing azetidinone analogs

US5759865A · kind A · utility

29Cited by
1References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 3, 1995
Grant dateJun 2, 1998
Priority date
Expiry dateMay 3, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC40B40/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to a combinatorial process for synthesizing a library of azetidinone peptide-like compounds. The compounds are synthesized as mixtures from a common azetidinone intermediate. The compounds are biologically active as inhibitors of the Vasopressin (V1a) receptor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.