Patent · US Expired

Preparation of optically-active isomers of dideoxycarbocyclic nucleosides

US5763607A · kind A · utility

4Cited by
19References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 10, 1996
Grant dateJun 9, 1998
Priority date
Expiry dateOct 10, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D473/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A method is provided for preparing an antiviral compound of formula (I): ##STR1## wherein Y is CH, Z is H or NH.sub.2, and X is halo, comprising: (a) reacting a compound of formula (II): ##STR2## with triethylorthoformate, and (b) hydrolyzing the product of said reaction in the presence of acid to yield said compound of formula (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.