Patent · US Expired

Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides

US5780590A · kind A · utility

5Cited by
13References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 21, 1996
Grant dateJul 14, 1998
Priority date
Expiry dateAug 21, 2016

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention is directed to a non-hygroscopic stable crystalline form of the antithrombotic compound N-N-N-(4-piperdin-4-yl)butanoyl)-N-ethylglycyl!-(L)-aspartyl!-(L)-.beta. -cyclohexyl-alanine amide, to processes for preparing said stable crystalline form, to a pharmaceutical composition thereof, and intermediates thereof, and the invention is directed also to processes for preparing a compound of the formula ##STR1## wherein: A, B, Z, E.sup.1, E.sup.2, G, R, m, n, and p are as defined herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.