Patent · US Expired

Guanidino protease inhibitors

US5792769A · kind A · utility

25Cited by
4References
49Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 15, 1996
Grant dateAug 11, 1998
Priority date
Expiry dateAug 15, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D211/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula: ##STR1## wherein R.sup.1 --R.sup.4, R.sup.7 --R.sup.8, R.sup.a, R.sup.b, R.sup.c, Y, Z, n and m are set forth in the specification, as well as hydrates, solvates or pharmaceutically acceptable salts thereof, that inhibit a number of proteolytic enzymes are described. Also described are methods for preparing the compounds of Formula I.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.