Patent · US Expired

Arteminolide derivatives and process for the manufacture thereof

US5801254A · kind A · utility

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3Claims
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Assignee

Inventors

Key dates

Filing dateAug 5, 1997
Grant dateSep 1, 1998
Priority date
Expiry dateAug 5, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D493/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Arteminolides obtained from Artemisia sylvatica MAXIMOWICZ and having a core structure of formula (I) or an isomeric structure thereof are effective farnesyl-protein transferase inhibitors as well as angiogenesis suppressors, and, accordingly, they are useful for the treatment of various cancers and angiogenesis-related diseases. ##STR1##

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.