Patent · US Expired

Process for the preparation of an intermediate useful in the synthesis of iodinated contrast media

US5817861A · kind A · utility

1Cited by
1References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 21, 1997
Grant dateOct 6, 1998
Priority date
Expiry dateMar 21, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C237/46
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process for the preparation of (S)-N,N'-bis2-hydroxy-1-(hydroxymethyl)ethyl!-5-(2-acetoxy-propionylamino )-2,4,6-triiodo-isophthalamide, an intermediate useful for the synthesis of iopamidol, by reaction between L-5-(2-acetoxy-propionylamino)-2,4,6-triiiodoisophthaloyl dichloride and 2-amino-1 ,3-propanediol in N-methylpyrrolidone and in the presence of a base, is described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.