Patent · US Expired

Branched hydrazone linkers

US5824805A · kind A · utility

167Cited by
27References
13Claims
0Family size

Inventors

Key dates

Filing dateDec 19, 1996
Grant dateOct 20, 1998
Priority date
Expiry dateDec 19, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H15/252
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Branched hydrazone linkers for linking a targeting ligand such as an antibody to a therapeutically active drug. The point of branching is at a polyvalent atom and the number of drugs increases by a factor of two for each generation of branching. A preferred drug is doxorubicin.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.