Patent · US Expired

Multivalent and multispecific binding proteins, their manufacture and use

US5837242A · kind A · utility

301Cited by
6References
85Claims
0Family size

Assignees

Inventors

Key dates

Filing dateMay 14, 1996
Grant dateNov 17, 1998
Priority date
Expiry dateMay 14, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12N2310/127
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Polypeptides comprising a first domain, which comprises a binding region of an immunoglobulin heavy chain variable region, and a second domain, which comprises a binding region of an immunoglobulin light chain variable region, the domains being linked but incapable of associating with each other to form an antigen binding site, associate to form antigen binding multimers, such as dimers, which may be multivalent or have multispecificity. The domains may be linked by a short peptide linker or may be joined directly together. Bispecific dimers may have longer linkers. Methods of preparation of the polypeptides and multimers and diverse repertoires thereof, and their display on the surface of bacteriophage for easy selection of binders of interest, are disclosed, along with many utilities.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.