Patent · US Expired

Triazole intermediates for tricyclic benzazepine and benzothiazepine derivatives

US5840895A · kind A · utility

15Cited by
2References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 26, 1997
Grant dateNov 24, 1998
Priority date
Expiry dateJun 26, 2017

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formulae (II), (III), (IV) and (V) or salts thereof are intermediates for pharmacologically active tricyclic benzazepine and benzothiazepine derivatives, ##STR1## wherein R represents hydrogen, alkyl, phenylalkyl, or a protective group of a triazole ring, R.sup.1 -R.sup.5 represent hydrogen, alkyl, alkenyl, alkoxy, amino, oxim or hydroxyl, and R.sup.41 represents hydrogen, C.sub.1-6 alkyl which may be optionally substituted, or a protective group for a carboxyl group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.