Patent · US Expired

Aromatic pyrrolidine amide prolyl endopeptidase inhibitors

US5847155A · kind A · utility

1Cited by
5References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 26, 1996
Grant dateDec 8, 1998
Priority date
Expiry dateJan 26, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D493/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A series of aromatic pyrrolidine derivatives and suitable pharmaceutically acceptable salts thereof are disclosed. These compounds are useful as PEP inhibitors in the treatment of Alzheimer's disease, amnesia, dementia, anxiety ischemia, or stroke.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.