Patent · US Expired

Arylheteroaryl inhibitors of farnesyl-protein transferase

US5859035A · kind A · utility

53Cited by
5References
31Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 27, 1997
Grant dateJan 12, 1999
Priority date
Expiry dateMar 27, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to compounds which inhibit famesyl-protein transferase (FTase) and the farnesylation of the oncogene protein Ras. The invention is further directed to chemotherapeutic compositions containing the compounds of this invention and methods for inhibiting famesyl-protein transferase and the famesyl of the oncogene protein Ras.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.