Synthesis of substituted N-heteroaromatic compounds and methods of use thereof
US5886186A · kind A · utility
5Cited by
7References
21Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Oct 25, 1995 |
| Grant date | Mar 23, 1999 |
| Priority date | — |
| Expiry date | Oct 25, 2015 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC40B40/00
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The subject invention features substituted N-heteroaromatic compounds, libraries of substituted N-heteroaromatic compounds, and methods of synthesis thereof. For example, the present invention provides methods for synthesizing substituted N-heteroaromatic compounds, and is particularly amenable to the generation of libraries of substituted N- heteroaromatic compounds by combinatorial chemistry. The methods of the invention generally feature the reaction of O-linked heteroaromatic N-oxides with nucleophiles to produce substituted N-heteroaromatic compounds.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.