Patent · US Expired

Serine protease inhibitor analogs

US5900400A · kind A · utility

6Cited by
24References
37Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 29, 1994
Grant dateMay 4, 1999
Priority date
Expiry dateJul 29, 2014

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10S530/854
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Analogs of the serine protease inhibitors in which the amino acid sequence is varied slightly are disclosed, which analogs variously show improved properties including improved resistance to oxidative inactivation, improved ability to inhibit pancreatic elastase, improved ability to inhibit cathepsin G, and improved ability to inhibit trypsin.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.