Patent · US Expired

Process for the preparation of roquinimex

US5912349A · kind A · utility

24Cited by
1References
6Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJan 13, 1998
Grant dateJun 15, 1999
Priority date
Expiry dateJan 13, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D215/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is an improved process to prepare roquinimex (IV) which comprises: PA1 (1) contacting N-methyl-N-phenyl-.alpha.-carbomethoxyamide (V) with from about one to about two equivalents of base and PA1 (2) contacting the mixture of step (1) with N-methylisatoic anhydride (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.