Patent · US Expired

Potassium ion channel blockers

US5929082A · kind A · utility

13Cited by
0References
15Claims
0Family size

Assignees

Inventors

Key dates

Filing dateJan 23, 1998
Grant dateJul 27, 1999
Priority date
Expiry dateJan 23, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D521/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention provides novel sulphonylurea, sulphonylthiourea and sulphonylguanidine compounds which have the ability to block potassium ion channels regulated by intracellular concentrations of ATP. Methods of synthesis, pharmaceutical compositions and methods for the treatment of conditions such as type II diabetes, cardiac arrhythmias, ischaemic and hypoxic cardiovascular incidents, and cancers are also claimed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.