Patent · US Expired

Process for preparation of 3-piperazinylbenzisothiazoles

US5939548A · kind A · utility

0Cited by
4References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 4, 1998
Grant dateAug 17, 1999
Priority date
Expiry dateAug 4, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D275/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

There is disclosed a process for preparing 3-piperazinylbenzisothiazoles comprising reacting the specified 3-halo-1,2-benzisothiazole or 2-cyanobenzenesulfenyl halide in the presence of an alkylene glycol derivative. The process is industrially effective, easy and economical and can provide useful intermediates for production of pharmaceutical preparations.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.