Patent · US Expired

Bicyclic oxazine and thiazine oxazolidinone antibacterials

US5952324A · kind A · utility

15Cited by
3References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 14, 1997
Grant dateSep 14, 1999
Priority date
Expiry dateMay 14, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Phenyloxazolidinone compound of formula (I)or a pharmaceutically acceptable salt thereof characterized by a bicyclic thiazine or oxazine substituent. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms such as Bacteroides spp. and Clostridia spp. species, and acid-fast organisms such as Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.