Cyclopentene derivatives useful as antagonists of the motilin receptor
US5972939A · kind A · utility
15Cited by
1References
9Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Oct 26, 1998 |
| Grant date | Oct 26, 1999 |
| Priority date | — |
| Expiry date | Oct 26, 2018 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07C2601/14
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The compounds of formula I are useful in treating gastrointestinal disorders associated with antagonizing the motilin receptor disorders. The compounds compete with erythromycin and motilin for the motilin receptor. In addition the compounds are antagonists of the contractile smooth muscle response to those ligands.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.