Patent · US Expired

Neuroprotective pharmaceutical composition containing stereoisomers of arylcyclohexylamines

US5972952A · kind A · utility

3Cited by
4References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 10, 1996
Grant dateOct 26, 1999
Priority date
Expiry dateDec 10, 2016

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/445
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to pharmaceutical compositions for neuroprotection containing the compound (1S,2R) 1-[1-(2-thienyl)-2-alkylcyclohexyl]piperidine or (1S,2R) 1-[1-(2-furanyl)-2-alkylcyclohexyl]piperdine, or their pharmaceutically acceptable salts. The synthesis and method separation of racemic mixtures to provide pure enantiomers is presented. The compositions have use in the treatment of stroke, CNS trauma and Alzheimer's disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.