Patent · US Expired

Dihydrobenzopyran compounds and related compounds useful as anti-inflammatory agents

US5972957A · kind A · utility

10Cited by
1References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 9, 1998
Grant dateOct 26, 1999
Priority date
Expiry dateApr 9, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound having the structure: ##STR1## wherein (a) n is from about 1 to about 3; PA1 (b) X is selected from the group consisting of O, S, SO, or SO.sub.2 ; PA1 (c) Y is independently hydrogen or straight, branched or cyclic alkyl having from 1 to about 4 carbon atoms, or the Y's are bonded together to form an alkanyl ring having from about 3 to about 7 atoms; PA1 (d) Z is hydrogen or straight, branched or cyclic alkyl having from 3 to about 10 atoms other than hydrogen; and PA1 (e) Het is a heteroaryl group comprising one or more rings each ring containing from about 5 to about 6 atoms other than hydrogen and wherein the group contains at least one heteroatom selected from O, N, or S. Pharmaceutical compositions comprising such compounds, and methods of treating inflammation or pair using such compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.