Patent · US Expired

Crystals of benzimidazole derivatives and their production

US6002011A · kind A · utility

22Cited by
1References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 21, 1998
Grant dateDec 14, 1999
Priority date
Expiry dateJan 21, 2018

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A substantially solvent-free and stable crystal of the compound of the formula: ##STR1## wherein the ring A may optionally be substituted, R.sup.1 represents hydrogen or an N-protecting group, each of R.sup.2, R.sup.3 and R.sup.4 (1) a hydrogen atom, (2) an alkyl group which may optionally be substituted with halogen atom(s) or (3) an alkoxy group which may optionally be substituted with halogen atom(s) or alkoxy; or its salt, is produced by subjecting a solvate of the compound (I) or its salt to de-solvent treatment, in an industrially advantageous method.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.