Patent · US Expired

Benzimidazole, benzoxazole and benzothiazole compounds

US6040327A · kind A · utility

17Cited by
1References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 22, 1998
Grant dateMar 21, 2000
Priority date
Expiry dateJul 22, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound of formula (I): ##STR1## wherein: R.sub.1 represents halogen or a different group as defined in the description, PA1 Ra and Rb, which mnay be identical or different, represent hydrogen, alkyl, or hydroxy, PA1 X represents oxygen or sulphur or NR, R being H or alkyl, PA1 R.sub.2 represents optionally-substituted aryl, PA1 R'.sub.2 represents hydrogen or optionally-substituted aryl, its isomers and addition salts thereof with a pharmaceutically-acceptable acid or base, and medicinal products containing the same, are useful as inhibitors of interleukin 1.beta..

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.