Patent · US Expired

Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritis therewith

US6054445A · kind A · utility

20Cited by
9References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 7, 1999
Grant dateApr 25, 2000
Priority date
Expiry dateMay 7, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided. The compound of formulae IIA, having the structure: ##STR1## wherein R.sub.1, R.sub.2 ; PA1 X.sub.4, X.sub.5 ; and PA1 Ar and n are as described in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.