Patent · US Expired

Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritus therewith

US6057323A · kind A · utility

21Cited by
12References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 30, 1998
Grant dateMay 2, 2000
Priority date
Expiry dateOct 30, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided. The compound of formula I, having the structure: ##STR1## wherein R.sub.1, R.sub.2 ; PA1 X; and Ar PA1 Y, Z and n are as described in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.