Patent · US Expired

Desformoterol compositions useful for inducing bronchodilation

US6071971A · kind A · utility

15Cited by
0References
10Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 5, 1999
Grant dateJun 6, 2000
Priority date
Expiry dateMay 5, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/07
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The (R,R)-, (S,S)-, (R,S)-, (R,S)-isomers of 3-amino-4-hydroxy-.alpha.-[[[2-(4-methoxyphenyl)-1-methylethyl]amino]methy l]-benzenemethanol (D) ##STR1## are disclosed, as well as an efficient method for their stereoselective synthesis. A method and composition are also disclosed utilizing desformoterol (D) as a bronchodilator, having high selectivity for .beta..sub.2 receptors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.