Patent · US Expired

Process to produce a protease inhibitor

US6077963A · kind A · utility

4Cited by
0References
45Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 17, 1998
Grant dateJun 20, 2000
Priority date
Expiry dateDec 17, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed is a novel process and novel intermediates to prepare [R-(R*,R*)]-N-[3-[1-[5,6-dihydro-4-hydroxy-2-oxo-6-(2-phenylethyl)-6-propy l-2H-pyran-3-yl]propyl]phenyl]-5-(trifluoromethyl)-2-pyridinesulfonamide (XIX) ##STR1## which is a protease inhibitor useful in treating humans infected with the HIV virus.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.