Patent · US Expired

Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides

US6080767A · kind A · utility

59Cited by
1References
43Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 27, 1997
Grant dateJun 27, 2000
Priority date
Expiry dateJun 27, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2603/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The compounds according to the invention are substituted N-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides of formula I herein which exhibit useful pharmacological activity and accordingly are incorporated into pharmaceutical compositions and used in the treatment of patients suffering from certain medical disorders. More especially, they are Factor Xa inhibitors. The present invention is directed to compounds of formula I, compositions containing compounds of formula I, methods for their preparation and their use, which are for treating a patient suffering from, or subject to, conditions which can be ameliorated by the administration of an inhibitor of Factor Xa.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.