Patent · US Expired

Compositions and methods for stimulating bone growth

US6080779A · kind A · utility

23Cited by
5References
20Claims
0Family size

Assignees

Inventors

Key dates

Filing dateJun 12, 1998
Grant dateJun 27, 2000
Priority date
Expiry dateJun 12, 2018

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/366
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## wherein X in each of formulas (1) and (2) represents a substituted or unsubstituted alkylene, alkenylene, or alkynylene linker of 2-6 C; Y represents one or more carbocyclic or heterocyclic rings; when two or more rings are present in Y, they may optionally be fused; and R' represents a cation, H or a substituted or unsubstituted alkyl group of 1-6 C; and the dotted lines represent optional .pi.-bonds, promote bone formation and are thus useful in treating osteoporosis, bone fracture or deficiency, primary or secondary hyperparathyroidism, periodontal disease or defect, metastatic bone disease, osteolytic bone disease, post-plastic surgery, post-prosthetic joint surgery, and post-dental implantation. These compounds can be used in combination with other bone growth-promoting compounds and/or estrogens and/or bisphosphonates for this purpose.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.