Patent · US Expired

8-azabicyclo[3.2.1.]oct-2-ene derivatives, their preparation and use

US6100275A · kind A · utility

1Cited by
7References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 18, 1998
Grant dateAug 8, 2000
Priority date
Expiry dateMay 18, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D451/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound having the formula, ##STR1## or any of its enantiomers or any mixture thereof, or a pharmaceutically acceptable salt thereof; PA0 wherein PA1 R is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl or 2-hydroxyethyl; and PA1 R.sup.4 is PA2 phenyl which may be substituted one or more times with substituents selected from the group consisting of halogen, CF.sub.3, CN, alkoxy, cycloalkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, amino, nitro, heteroaryl and aryl; PA2 3,4-methylenedioxyphenyl; PA2 benzyl which may be substituted one or more times with substituents selected from the group consisting of halogen, CF.sub.3, CN, alkoxy, cycloalkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, amino, nitro, heteroaryl and aryl; PA2 heteroaryl which may be substituted one or more times with substituents selected from the group consisting of halogen, CF.sub.3, CN, alkoxy, cycloalkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, amino, nitro, heteroaryl and aryl; or PA2 naphthyl which may be substituted one or more times with substituents selected from the group consisting of halogen, CF.sub.3, CN, alkoxy, cycloalkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, amino, nitro, heteroaryl and aryl…

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.