Patent · US Expired

Systems and methods for topical treatment with nitric oxide

US6103275A · kind A · utility

277Cited by
17References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 10, 1998
Grant dateAug 15, 2000
Priority date
Expiry dateJun 10, 2018

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A simple, biocompatible system and procedure for generating nitric oxide (NO) is described. A mixture of powdered sodium nitrite, ascorbic acid, and maleic acid (or another organic acid of adequate strength) immediately generates nitric oxide (NO) on treatment with water. To slow down the NO generation, one may prepare an ointment from a nonaqueous medium (petrolatum, vaseline) and the three powdered ingredients, which on being applied topically on the skin will release NO as water permeates through this medium; alternatively, one may convert the aqueous sodium nitrite solution into a gel with hydroxyethylcellulose (or other gel-forming compound) and combine this gel with another gel obtained from aqueous ascorbic and maleic acids with hydroxyethylcellulose for topical application (on intact skin, burns, intra-cavity, etc.). The two gels may be admixed immediately before use (possibly from a single container with separate chambers and dual nozzle, via pushing or squeezing the two gels through the nozzle), or may be applied in sandwich-like fashion (possibly as a transdermal patch) for further slowing down the delivery of NO.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.