Patent · US Expired

N-aryloxyethylamine derivatives for the treatment of depression

US6110956A · kind A · utility

2Cited by
3References
35Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 7, 1999
Grant dateAug 29, 2000
Priority date
Expiry dateApr 7, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds effective in treating disorders of the serotonin-affected neurological systems are provided, such compounds having the following formula: ##STR1## wherein: R.sub.1 and R.sub.2 are each, independently, hydrogen, halogen, CF.sub.3, lower alkyl, lower alkoxy, MeSO.sub.2, or together can form a 5-7 membered carbocyclic or heterocyclic ring; PA1 R.sub.3 is alkoxy, halogen, hydrogen or carbamoyl; PA1 R.sub.4 is hydrogen, hydroxy, lower alkyl, or lower alkoxy; PA1 R.sub.5 is hydrogen, lower alkyl, or halogen; PA1 R.sub.6 is hydrogen, lower alkyl, or phenyl; PA1 R.sub.7 is hydrogen, lower alkyl, lower alkoxy, halogen, CN, CF.sub.3, or hydroxy; and PA1 X is (CH.sub.2).sub.n, PA1 wherein n is 0 to 3; or pharmaceutically acceptable salts thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.