Pyrimido[1,2-a]indoles

US6114341A · kind A · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Ulrich Muller · Wuppertal, DE
• Peter Eckenberg · Wuppertal, DE
• Rudi Grutzmann · Solingen, DE
• Hilmar Bischoff · Wuppertal, DE
• Dirk Denzer · Wuppertal, DE
• Stefan Wohlfeil · Hilden, DE
• Stefan Lohmer · Milano, IT
• Ulrich Nielsch · Wuppertal, DE
• Peter Kolkhof · Wuppertal, DE

Key dates

• Filing date: Mar 31, 1997
• Grant date: Sep 5, 2000
• Expiry date: Mar 31, 2017

Classification

• Technology area (CPC A): Human Necessities
• CPC primary: A61P9/10
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

The pyrimido[1,2-a]indoles according to the invention are prepared by reacting appropriately substituted phenylacetic acid derivatives with phenylglycinols. The pyrimido[1,2-a]indoles can be used as active compounds in medicaments, in particular in medicaments with antiatherosclerotic activity.