Patent · US Expired

Substituted phenols and thiophenols useful as antioxidant agents

US6114572A · kind A · utility

3Cited by
45References
32Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 19, 1997
Grant dateSep 5, 2000
Priority date
Expiry dateNov 19, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C323/20
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of the formula ##STR1## wherein X is selected from the group consisting of ##STR2## Y is thio, oxy or a methylene group; Z is hydrogen or --C(O)--(CH.sub.2).sub.m --Q wherein Q is hydrogen or --COOH and m is an integer 1, 2, 3 or 4; PA1 R.sub.1 is C.sub.1 -C.sub.6 alkyl; and PA1 R.sub.2, R.sub.3 and R.sub.4 are each independently hydrogen or C.sub.1 -C.sub.6 alkyl; or a stereoisomer thereof; useful for the treatment of atherosclerosis and chronic inflammatory disorders; for inhibiting cytokine-induced expression of VCAM-1 and/or ICAM-1; for inhibiting the peroxidation of LDL lipid; for lowering plasma cholesterol; and as anti-oxidant chemical additives useful for preventing oxidative deterioration in organic materials.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.