Patent · US Expired

Substituted aminoalkane phosphonic acids

US6117873A · kind A · utility

23Cited by
6References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 23, 1999
Grant dateSep 12, 2000
Priority date
Expiry dateApr 23, 2019

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula I ##STR1## in which R.sub.1 is hydroxyl or an aliphatic, araliphatic or aromatic radical, PA1 X is a divalent aliphatic, cycloaliphatic, cycloaliphatic-aliphatic, araliphatic, heteroarylaliphatic or aromatic radical, PA1 R.sub.2 is hydrogen or an aliphatic or araliphatic radical, alk is lower alkylidene and PA1 R.sub.3, R.sub.4 and R.sub.5 independently of one another are hydrogen, lower alkyl, halogen, trifluoromethyl, cyano or nitro, and their salts can be used for the treatment of pathological conditions which respond to blockage of excitatory amino acid receptors, and for the production of pharmaceutical preparations.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.