Patent · US Expired

Stable oral CI-981 formulation and process for preparing same

US6126971A · kind A · utility

25Cited by
3References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 2, 1997
Grant dateOct 3, 2000
Priority date
Expiry dateJul 2, 2017

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/40
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An oral pharmaceutical composition is provided for treating hypercholestereolemia or hyperlipidemia containing an advantageous formulation for stabilizing the HMG-CoA coenzyme A inhibitor, CI-981 Hemi-Calcium, of formula (IA) ##STR1## with effective amounts of calcium carbonate. A method for preparing a CI-981 stabilizing composition is described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.