Patent · US Expired

Morpholino-n-ethyl ester derivative of an indole sPLA.sub.2 inhibitor

US6140327A · kind A · utility

1Cited by
1References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 12, 1999
Grant dateOct 31, 2000
Priority date
Expiry dateMay 12, 2019

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The compound, ((3-(2-amino-1,2-dioxoethyl)-2-ethyl-1-(phenylmethyl)-1H-indol-4-yl)oxy)ac etic acid morpholino-N-ethyl ester, is disclosed together with its use as a highly bioavailable indole compound for inhibiting sPLA.sub.2 mediated release of fatty acids for treatment of conditions such as septic shock.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.