Patent · US Expired

Method for preparation of disodium pamidronate

US6160165A · kind A · utility

1Cited by
25References
7Claims
0Family size

Assignee

Inventor

Key dates

Filing dateDec 10, 1998
Grant dateDec 12, 2000
Priority date
Expiry dateDec 10, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/3873
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention includes a method for the preparation of disodium pamidronate comprising: (a) preparing a stirred slurry of pamidronate in water, (b) adding a solution of sodium hydroxide to give a clear solution at pH of about 6.5, (c) filtering the solution and (d) freezing and lyophilizing the solution to give an amorphous essentially anhydrous disodium pamidronate which contains .ltoreq.2 wt-% water.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.