Patent · US Expired

3,4-diamino-3-cyclobutene-1,2-dione derivatives which inhibit leukocyte adhesion mediated by VLA-4

US6166050A · kind A · utility

27Cited by
1References
39Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 10, 1999
Grant dateDec 26, 2000
Priority date
Expiry dateDec 10, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## which inhibit leukocyte adhesion mediated by interaction of the .alpha..sub.4 .beta..sub.1 integrin (VLA-4) with its counterreceptor VCAM-1, and their use for the treatment of inflammatory and autoimmune diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.