Patent · US Expired

Dihydropyrimidines and uses thereof

US6172066A · kind A · utility

11Cited by
21References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 16, 1997
Grant dateJan 9, 2001
Priority date
Expiry dateMay 16, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D239/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention is directed to dihydropyrimidine compounds which are selective antagonists for human .alpha..sub.1A receptors. This invention is also related to uses of these compounds for lowering intraocular pressure, inhibiting cholesterol synthesis, relaxing lower urinary tract tissue, the treatment of benign prostatic hyperplasia, impotency, cardiac arrhythmia and for the treatment of any disease where the antagonism of the .alpha..sub.1A receptor may be useful. The invention further provides a pharmaceutical composition comprising a therapeutically effective amount of the above-defined compounds and a pharmaceutically acceptable carrier.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.