Patent · US Expired

Composition and methods employing it for the treatment of 5-HT-mediated disorders

US6172105A · kind A · utility

4Cited by
1References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 9, 1999
Grant dateJan 9, 2001
Priority date
Expiry dateJul 9, 2019

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P25/26
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to a composition comprising a first component (a) which is (R)-3-N,N-dicyclobutylamino-8-fluoro-3,4-dihydro-2H-1-benzopyran-5-carboxa mide hydrogen (2R,3R)-tartrate monohydrate and a second component (b) which is a 5-HT reuptake inhibitor, excluding citalopram and paroxetine. The invention is further directed to the preparation of the composition, pharmaceutical formulations containing said composition, and a method of treatment of affective disorders such as mood disorders and anxiety disorders with said composition, as well as a kit containing said composition.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.