Patent · US Expired

Spirodiamino acid scaffold for combinatorial synthesis

US6175020A · kind A · utility

0Cited by
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12Claims
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Assignee

Inventors

Key dates

Filing dateApr 9, 1999
Grant dateJan 16, 2001
Priority date
Expiry dateApr 9, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D209/54
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Azaspirononanes of formula I and their synthesis ##STR1## are disclosed. The compounds are useful as templates for constructing synthetic receptors and as intermediates in the synthesis of enzyme inhibitors. They are prepared by an intramolecular ylide cycloaddition of a 6-hydrazone of 2,10-undecadienoic acid ester.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.